Bisnortilidine

Bisnortilidine
Names

IUPAC name Ethyl (1R,2S)-2-amino-1-phenylcyclohex-3-ene-1-carboxylate
Identifiers
3D model (Jmol)	Interactive image
ChemSpider	454879
PubChem	162740
InChI InChI=1S/C15H19NO2/c1-2-18-14(17)15(11-7-6-10-13(15)16)12-8-4-3-5-9-12/h3-6,8-10,13H,2,7,11,16H2,1H3/t13-,15+/m0/s1 Key: BTKAMSWFNMGLGM-DZGCQCFKSA-N
SMILES CCOC(=O)[C@]1(CCC=C[C@@H]1N)C2=CC=CC=C2
Properties
Chemical formula	C₁₅H₁₉NO₂
Molar mass	245.32 g·mol⁻¹
Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa).
Infobox references

Bisnortilidine is an opioid metabolite.^[1] It is formed from tilidine by demethylation in the liver.

References

↑ Wustrow, I.; Riedel, K. D.; Mikus, G.; Weiss, J. (2012). "In vitro identification of the cytochrome P450 isozymes involved in the N-demethylation of the active opioid metabolite nortilidine to bisnortilidine". Naunyn-Schmiedeberg's Archives of Pharmacology. 385 (6): 633–9. doi:10.1007/s00210-012-0737-z. PMID 22349139.

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